1.前药分子设计进展（Advance in Prodrug Design）&郭宗儒 1
2.药物手性及其生物活性（Chirality and the Biological Activity of Drugs）&华维一 18
3.血小板凝集抑制剂研究进展（Progress in Platellt Inhibitors）&黄枕亚 39
4.非常规精神病药物研究进展（Progress in Atypical Antipsychotic Agents）&嵇汝运 70
5.可逆乙酰胆碱酯酶抑制剂分子模型和定量构效关系（Molecular Model of Revorse Acetylcholinesterase Inhibiters and Their QSAR）&张明强 林克江 尤启冬 88
6.整合素及以之为靶的药物（Integrins and Drugs Acting on It as Target）&彭师奇 111
7.抗哮喘药物研究进展（Progress in Asthma Drug Discovery）&王鹏 133
8.β-内酰胺类抗生素研究的进展（Progress in Research ofβ-Lactam Antibiotics）&张致平 166
9.肿瘤多药耐药机制及其逆转新策略（The Mechanisms and New Reversal Strategies on Multidrug Resistance of Cancer Cell）&杨纯正 彭晖 王树滨 181
10.抗体导向的酶-前药治疗肿瘤的研究（Study on Antibody Directed Enzyme-Prodrug Therapy for Cancer）&王艺 尤启冬 207
11.脑缺血和神经元保护剂（Cerebral Ischemia and Neuroprotective Agents）&刘国卿 225
12.环氧酶-2及其选择性抑制剂的研究进展（Progress in Cyclooxygenase-2 and its Selective Inhibitors）&敖桂珍 张奕华 张玉彬 237
13.羟甲基戊二酰辅酶A（HMG-CoA）还原酶抑制剂研究进展（Recent Development of Hydroxymethylglutaryl Coenzyme A Reductase Inhibitor）&黄文龙 张惠斌 248
14.天然产物分离和结构研究技术的新进展（Recent Advances in Isolation and Structural Research of Nature Products）&孔令义 郑训海 261
15.肝损伤动物模型与药效评价（Animal Models of Liver Injury for the Evaluation of Remedies for Hepatitis）&徐强 277
16.从天然产物中寻找神经生长因子诱导剂（The Nerve Growth Factor Induces from Natural Products）&闵知大 王朝虹 梁侨丽 291
索引 303