承师创新 3
李正名简历 3
李正名自述 5
饮水思源——恩师杨石先先生对农药化学学科的重要贡献及其学术思想 9
业绩与奖项 16
主要科研项目 18
论文选登 23
1957年 23
萘和苯的衍生物类生长素对植物插枝生根作用的初步报告 23
1959年 35
有机磷杀虫剂的研究Ⅰ 35
1962年 44
有机磷杀虫剂的研究Ⅱ 44
1963年 48
有机磷杀虫剂的研究Ⅲ 48
1965年 54
有机磷杀虫剂的研究Ⅶ 54
1983年 63
UV-Ozonation and Land Disposal of Aqueous Pesticide Wastes 63
内吸杀菌剂三唑醇立体异构体研究初报 69
1984年 73
棉铃虫拟信息素正十四烷基甲酸酯及有关化合物的触角电位反应 73
A Convenient Synthetic Route for the Sex Pheromone of the Asian Corn Borer Moth(Ostrinia furnacalis Guenee) 76
1987年 83
内吸性杀菌剂三唑醇(酮)立体异构体的研究(Ⅱ) 83
1-(4-氯苯氧基-3,3-二甲基-1-(1,2,4-三氮唑-1基)-丁醇2右旋A体的晶体结构和绝对构型 89
1989年 93
A Stereoselective Synthesis of Pear Ester via Arsenic Ylide 93
1990年 96
The Chemical Characterization of the Cephalic Secretion of the Australian Colletid Bee,Hylaeus albonitens(Gnathoprosopls Cockerell) 96
The Wittig Sigmatropic Rearrangement in a Conjugated Diene System Ⅰ 105
山梨酸的合成及其生物活性研究 111
1991年 120
茶尺蠖性信息素化学结构研究初报 120
1992年 123
新磺酰脲类化合物的合成、结构及构效关系研究(Ⅰ) 123
1993年 129
新磺酰脲类化合物的合成、结构及构效关系研究(Ⅱ) 129
Structural Elucidation of Sex Pheromone Components of the Geometridae Semiothisa cinerearia(Bremer et Grey)in China 134
1994年 140
新磺酰脲类化合物的合成、结构及构效关系研究(Ⅲ) 140
The Reaction of α-oxo-α-Triazolylketene Dithioacetal with Amines,Hydrazine and Guanidine 144
Studies on Sex Pheromone of Ectropis obliqua Prout 147
1995年 155
Synthesis of 5-Mercaptoalkylamino-and 5-Anilinoalkylthiopyrazolyl-1,2,4-Triazoles by Ring Chain Transformation 155
1996年 161
Synthesis and base-catalyzed Protodesilylation of 5-(Silylmethylthio)-3(2H)-Pyridazinone Derivatives 161
Synthesis of 5-mercaptoalkylthiopyrazolyl-and3-mercaptoalkyl thioisoxazolyl-1,2,4-triazoles by Ring Chain Transformation 168
1997年 172
新磺酰脲类化合物的合成、结构及构效关系研究(Ⅴ) 172
新型杀菌剂β-甲氧基丙烯酸甲酯类化合物的合成方法概述 176
1998年 182
3-吡唑基-6-取代均三唑并[3,4-b]-1,3,4-噻二唑的合成及生物活性 182
Syntheses of Di-heterocyclic Compounds;Pyrazolylimidazoles and Isoxazolylimidazoles 187
3-芳基磺酰氧基(取代)异噻唑的合成及除草活性 192
应用CoMFA研究磺酰脲类化合物的三维构效关系 197
2,5-二吡唑基-1,3,4-噁二唑的一锅煮法合成及生物活性 202
1999年 205
2-芳甲酰氨基硫羰基-3-异噻唑酮及4-氰基-5-甲硫基-2-芳甲酰氨基硫羰基-3-异噻唑酮的合成与生物活性 205
The Design and Synthesis of ALS Inhibitors from Pharmacophore Models 210
2000年 215
新磺酰脲类化合物的合成、结构及构效关系研究(Ⅵ) 215
Synthesis and Fungicidal Activity against Rhizoctonia solani of 2-Alkyl(Alkylthio)-5-pyrazolyl-1,3,4-oxadiazoles(Thiadiazoles) 220
2001年 229
N-(取代嘧啶-2′-基)-2-三氟乙酰氨基苯磺酰脲的合成及除草活性 229
新磺酰脲类除草活性构效关系的研究 233
2002年 240
卤代-2-(3-甲基-5-取代-4H-1,2,4-三唑-4-基)-苯甲酸的合成 240
5-依维菌素B1a酯的合成和生物活性 244
2-(1H-咪唑-1-基)-1-(2,3,4-三甲氧基)苯乙酮肟酯新化合物合成与生物活性研究 256
2003年 262
1,3-二甲基-5-甲硫基-4-苯腙基羰基吡唑的合成及抑菌活性 262
Metal Ion Interactions with Sugars.The Crystal Structure and FT-IR Study of the NdCl3-ribose Complex 266
3-Methylthio-pyrano[4,3-c]pyrazol-4(2H)-ones from 3-(Bis-methylthio)methylene-2H-pyran-2,4-diones and Hydrazines 277
2004年 281
新单取代苯磺酰脲衍生物的合成及生物活性 281
N-(4-取代嘧啶-2-基)苄基磺酰脲和苯氧基磺酰脲的3D-QSAR研究 287
基于酮醇酸还原异构酶KARI复合物晶体结构的三维数据库搜寻 291
N-杂环-3-N′-苄氧羰基-β-氨基丁酰胺的合成和结构表征 296
Synthesis and Biological Activity of Novel 2-Methyl-4-trifluoromethyl-thiazole-5-carboxamide derivatives 302
Metal-ion Interactions with Sugars Crystal Structures and FT-IR Studies of the LaCl3-ribopyranose and CeCl3-ribopyranose Complexes 308
2005年 324
一类新型嘧啶苯氧(硫)醚的合成及生物活性 324
4-(取代嘧啶-2-基)-1-芳磺酰基氨基脲化合物的合成与表征 331
Synthesis and Fungicidal Activity of Novel 2-Oxocycloalkylsulfonylureas 339
Synthesis,Crystal Structure and Herbicidal Activity of Mimics of Intermediates of the KARI Reaction 349
Synthesis and Herbicidal Activity of 2-Alkyl(aryl)-3-methylsulfonyl(sulfinyl)pyrano-[4,3-c]pyrazol-4(2H)-ones 358
2006年 364
单嘧磺隆除草剂的晶体构象-活性构象转换的密度泛函理论研究 364
O-取代苯基-O-(2-硬脂酰胺基)乙基-N,N-二(2-氯乙基)磷酰胺的合成和生物活性 376
3-N-苄氧羰基-β-氨基丁酸水杨酸酯类化合物的合成及其生物活性 383
Synthesis and Crystal Structure of 5-N-i-Propyl-2-(2′-nitrobenzene-sulfonyl)-glutamine 389
Synthesis,Dimeric Crystal Structure,and Biological Activities of N-(4-Methyl-6-oxo-1,6-dinydro-pyrimidin-2-yl)-N′-(2-trifluoro-methyl-phenyl)-guanidine 394
Microwave and Ultrasound Irradiation-Assisted Synthesis of Novel Disaccharide-Derived Arylsulfonyl Thiosemicarbazides 400
2007年 406
Synthesis of New Plant Growth Regulator:N-(fatty acid)O-aryloxyacetyl Ethanolamine 406
Synthesis,Bioactivity,Theoretical and Molecular Docking Study of 1-Cyano-N-substituted-cyclopropanecarboxamide as Ketol-acid Reductoisomerase Inhibitor 411
单嘧磺隆晶体-活性构象转换的分子动力学模拟 420
基于受体结构的AHAS抑制剂的设计、合成及生物活性 427
The Design,Synthesis,and Biological Evaluation of Novel Substituted Purines as HIV-1 Tat-TAR Inhibitors 431
酵母AHAS酶与磺酰脲类抑制剂作用模型的分子对接研究 444
2008年 450
High Throughput Screening Under Zinc-Database and Synthesis a Dialkylphos-phinic Acid as a Potential Kari Inhibitor 450
N-(4′-取代嘧啶-2′-基)-2-甲氧羰基-5-(取代)苯甲酰胺基苯磺酰脲化合物的合成及除草活性研究 453
Synthesis and Herbicidal Activity of Novel Sulfonylureas Containing Thiadiazol Moiety 465
The Outset Innovation of Agrochemicals in China 471
2009年 477
Quantitive-structure Activity Relationship(QSAR)Study of a New Heterocyclic Insecticides Using CoMFA and CoMSIA 477
Design,Synthesis,and Fungicidal Activity of Novel Analogues of Pyrrolnitrin 483
新型苯环5-(取代)苯甲酰胺基苯磺酰脲类化合物的比较定量构效关系研究 496
Regioselective Synthesis of Novel 3-Alkoxy(phenyl)thiophosphorylamido-2-(per-O-acetylglycosyl-1′-imino) Thiazolidine-4-one Derivatives from O-alkyl N4-glycosyl(thiosemicarbazido) Phosphonothioates 501
Synthesis,Herbicidal Activities and Comparative Molecular Field Analysis Study of Some Novel Triazolinone Derivatives 512
Synthesis,Antifungal Activities and 31D-QSAR Study of N-(5-substituted-1,3,4-thiadiazol-2-yl) Cyclopropanecarboxamides 526
Synthesis,Bioactivity and SAR Study of N′-(5-substituted-1,3,4-thiadiazol-2-yl)-N-cyclopropylformyl-thioureas as Ketol-acidReductoisomerase Inhibitors 535
Synthesis and Biological Activity of Novel 2,3-Dihydro-2-phenylsulfonyl-hydrazono-3-(2′,3′,4′,6′-tetra-O-acetyl-β-D-glucopyranosyl)thiazoles 546
4,5,6-三取代嘧啶苯磺酰脲类化合物的生物活性、分子对接与3D-QSAR关系研究 552
2010年 559
Synthesis, Crystal Structure and Insecticidal Activities of Novel Neonicotinoid Derivatives 559
区域选择性合成2-取代磺酰基亚肼基-3-全乙酰糖基-2, 3-二氢噻唑及其表征、生物活性研究 567
3位苯甲酰腙和亚氨基取代硫脲取代的吲哚满二酮衍生物的合成及对AHAS的抑制活性 573
Synthesis and Biological Activity of Some Novel Trifluoromethyl-Substituted 1,2,4-Triazole and Bis(1,2,4-Triazole) Mannich Bases Containing Piperazine Rings 578
Synthesis and Fungicidal Activity of Novel Aminophenazine-1-carboxylate Derivatives 594
High Throughput Receptor-based Virtual Screening under ZINC Database,Synthesis,and Biological Evaluation of Ketol-acid Reductoisomerase Inhibitors 618
2011年 627
Synthesis and Insecticidal Activities of Novel Analogues of Chlorantraniliprole Containing Nitro Group 627
Modulations of High-voltage Activated Ca2+ Channels in the Central Neurones of Spodoptera Exigua by Chlorantraniliprole 634
Synthesis,Structure and Biological Activity of Novel 1,2,4-Triazole Mannich Bases Containing a Substituted Benzylpiperazine Moiety 641
Design,Synthesis and Antifungal Activities of Novel Pyrrole Alkaloid Analogs 654
Synthesis and Insecticidal Evaluation of Novel N-Pyridylpyrazolecarboxamides Containing Different Substituents in the ortho-Position 675
Synthesis,Crystal Structure,Bioactivity and DFT Calculation of New Oxime Ester Derivatives Containing Cyclopropane Moiety 684
2012年 693
The Structure-activity Relationship in Herbicidal Monosubstituted Sulfonylureas 693
Synthesis,Crystal Structure and Biological Activities of Novel Anthranilic ( Isoph-thalic)Acid Esters 708
Synthesis and Evaluation of Novel Monosubstituted Sulfonylurea Derivatives as Antituberculosis Agents 716
基于Ugi反应的新型鱼尼丁受体杀虫剂的设计、合成及生物活性 736
Synthesis and Insecticidal Activities of Novel Anthranilic Diamides Containing Acylthiourea and Acylurea 746
Design,Synthesis and Biological Activities of Novel Anthranilic Diamide Insecticide Containing Trifluoroethyl Ether 760
Evaluation of the in Vitro and Intracellular Effiicacy of New Monosubstituted Sulfonylureas against Extensively Drug-resistant Tuberculosis 779
2013年 786
Synthesis and Insecticidal Evaluation of Novel N-Pyridylpyrazolecarboxamides Containing Cyano Substituent in the ortho-Position 786
N-[4-氯-2-取代氨基甲酰基-6-甲基苯基]-1-芳基-5-氯-3-三氟甲基-1 H-吡唑-4-甲酰胺的合成及生物活性 795
Synthesis,Insecticidal Activities,and SAR Studies of Novel Pyridylpyrazole Acid Derivatives Based on Amide Bridge Modification of Anthranilic Diamide Insecticides 805
Design,Synthesis and Structure-activity of N-Glycosyl-1-pyridyl-1H- pyrazole-5-carboxamide as Inhibitors of Calcium Channels 826
新型含三唑啉酮的磺酰脲类化合物的合成、晶体结构及除草活性研究 839
Design,Syntheses and Biological Activities of Novel Anthranilic Diamide Insecticides Containing N-Pyridylpyrazole 853
Synthesis and Biological Activities of Novel Anthranilic Diamides Analogues Containing Benzo[b]thiophene 865
附录 879
附录1论文总目录 879
附录2专利及著作目录 911
附录3历年指导的学生名单 915