《李正名文集》PDF下载

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  • 作  者:《李正名文集》编委会编
  • 出 版 社:北京:冶金工业出版社
  • 出版年份:2014
  • ISBN:9787502464707
  • 页数:916 页
图书介绍:《李正名文集》将李正名院士及其科研团队自1957年至今所研究发表的学术论文,按照时间顺序和研究内容进行了整合编排,内容涉及农药与环境安全、农药合成、分析、毒理、抗性、应用等诸多领域。由于文章数量较多,本书从中选取了161篇有代表性的论文进行了全文收录,其他论文则只对题目、收录期刊以及发表时间进行整理。书稿中所有论文都已在不同的期刊上发表过,有些发表年代还较早,所以单位和量的表述方法基本忠实于原文,没有按现在的出版规范进行修改。

承师创新 3

李正名简历 3

李正名自述 5

饮水思源——恩师杨石先先生对农药化学学科的重要贡献及其学术思想 9

业绩与奖项 16

主要科研项目 18

论文选登 23

1957年 23

萘和苯的衍生物类生长素对植物插枝生根作用的初步报告 23

1959年 35

有机磷杀虫剂的研究Ⅰ 35

1962年 44

有机磷杀虫剂的研究Ⅱ 44

1963年 48

有机磷杀虫剂的研究Ⅲ 48

1965年 54

有机磷杀虫剂的研究Ⅶ 54

1983年 63

UV-Ozonation and Land Disposal of Aqueous Pesticide Wastes 63

内吸杀菌剂三唑醇立体异构体研究初报 69

1984年 73

棉铃虫拟信息素正十四烷基甲酸酯及有关化合物的触角电位反应 73

A Convenient Synthetic Route for the Sex Pheromone of the Asian Corn Borer Moth(Ostrinia furnacalis Guenee) 76

1987年 83

内吸性杀菌剂三唑醇(酮)立体异构体的研究(Ⅱ) 83

1-(4-氯苯氧基-3,3-二甲基-1-(1,2,4-三氮唑-1基)-丁醇2右旋A体的晶体结构和绝对构型 89

1989年 93

A Stereoselective Synthesis of Pear Ester via Arsenic Ylide 93

1990年 96

The Chemical Characterization of the Cephalic Secretion of the Australian Colletid Bee,Hylaeus albonitens(Gnathoprosopls Cockerell) 96

The Wittig Sigmatropic Rearrangement in a Conjugated Diene System Ⅰ 105

山梨酸的合成及其生物活性研究 111

1991年 120

茶尺蠖性信息素化学结构研究初报 120

1992年 123

新磺酰脲类化合物的合成、结构及构效关系研究(Ⅰ) 123

1993年 129

新磺酰脲类化合物的合成、结构及构效关系研究(Ⅱ) 129

Structural Elucidation of Sex Pheromone Components of the Geometridae Semiothisa cinerearia(Bremer et Grey)in China 134

1994年 140

新磺酰脲类化合物的合成、结构及构效关系研究(Ⅲ) 140

The Reaction of α-oxo-α-Triazolylketene Dithioacetal with Amines,Hydrazine and Guanidine 144

Studies on Sex Pheromone of Ectropis obliqua Prout 147

1995年 155

Synthesis of 5-Mercaptoalkylamino-and 5-Anilinoalkylthiopyrazolyl-1,2,4-Triazoles by Ring Chain Transformation 155

1996年 161

Synthesis and base-catalyzed Protodesilylation of 5-(Silylmethylthio)-3(2H)-Pyridazinone Derivatives 161

Synthesis of 5-mercaptoalkylthiopyrazolyl-and3-mercaptoalkyl thioisoxazolyl-1,2,4-triazoles by Ring Chain Transformation 168

1997年 172

新磺酰脲类化合物的合成、结构及构效关系研究(Ⅴ) 172

新型杀菌剂β-甲氧基丙烯酸甲酯类化合物的合成方法概述 176

1998年 182

3-吡唑基-6-取代均三唑并[3,4-b]-1,3,4-噻二唑的合成及生物活性 182

Syntheses of Di-heterocyclic Compounds;Pyrazolylimidazoles and Isoxazolylimidazoles 187

3-芳基磺酰氧基(取代)异噻唑的合成及除草活性 192

应用CoMFA研究磺酰脲类化合物的三维构效关系 197

2,5-二吡唑基-1,3,4-噁二唑的一锅煮法合成及生物活性 202

1999年 205

2-芳甲酰氨基硫羰基-3-异噻唑酮及4-氰基-5-甲硫基-2-芳甲酰氨基硫羰基-3-异噻唑酮的合成与生物活性 205

The Design and Synthesis of ALS Inhibitors from Pharmacophore Models 210

2000年 215

新磺酰脲类化合物的合成、结构及构效关系研究(Ⅵ) 215

Synthesis and Fungicidal Activity against Rhizoctonia solani of 2-Alkyl(Alkylthio)-5-pyrazolyl-1,3,4-oxadiazoles(Thiadiazoles) 220

2001年 229

N-(取代嘧啶-2′-基)-2-三氟乙酰氨基苯磺酰脲的合成及除草活性 229

新磺酰脲类除草活性构效关系的研究 233

2002年 240

卤代-2-(3-甲基-5-取代-4H-1,2,4-三唑-4-基)-苯甲酸的合成 240

5-依维菌素B1a酯的合成和生物活性 244

2-(1H-咪唑-1-基)-1-(2,3,4-三甲氧基)苯乙酮肟酯新化合物合成与生物活性研究 256

2003年 262

1,3-二甲基-5-甲硫基-4-苯腙基羰基吡唑的合成及抑菌活性 262

Metal Ion Interactions with Sugars.The Crystal Structure and FT-IR Study of the NdCl3-ribose Complex 266

3-Methylthio-pyrano[4,3-c]pyrazol-4(2H)-ones from 3-(Bis-methylthio)methylene-2H-pyran-2,4-diones and Hydrazines 277

2004年 281

新单取代苯磺酰脲衍生物的合成及生物活性 281

N-(4-取代嘧啶-2-基)苄基磺酰脲和苯氧基磺酰脲的3D-QSAR研究 287

基于酮醇酸还原异构酶KARI复合物晶体结构的三维数据库搜寻 291

N-杂环-3-N′-苄氧羰基-β-氨基丁酰胺的合成和结构表征 296

Synthesis and Biological Activity of Novel 2-Methyl-4-trifluoromethyl-thiazole-5-carboxamide derivatives 302

Metal-ion Interactions with Sugars Crystal Structures and FT-IR Studies of the LaCl3-ribopyranose and CeCl3-ribopyranose Complexes 308

2005年 324

一类新型嘧啶苯氧(硫)醚的合成及生物活性 324

4-(取代嘧啶-2-基)-1-芳磺酰基氨基脲化合物的合成与表征 331

Synthesis and Fungicidal Activity of Novel 2-Oxocycloalkylsulfonylureas 339

Synthesis,Crystal Structure and Herbicidal Activity of Mimics of Intermediates of the KARI Reaction 349

Synthesis and Herbicidal Activity of 2-Alkyl(aryl)-3-methylsulfonyl(sulfinyl)pyrano-[4,3-c]pyrazol-4(2H)-ones 358

2006年 364

单嘧磺隆除草剂的晶体构象-活性构象转换的密度泛函理论研究 364

O-取代苯基-O-(2-硬脂酰胺基)乙基-N,N-二(2-氯乙基)磷酰胺的合成和生物活性 376

3-N-苄氧羰基-β-氨基丁酸水杨酸酯类化合物的合成及其生物活性 383

Synthesis and Crystal Structure of 5-N-i-Propyl-2-(2′-nitrobenzene-sulfonyl)-glutamine 389

Synthesis,Dimeric Crystal Structure,and Biological Activities of N-(4-Methyl-6-oxo-1,6-dinydro-pyrimidin-2-yl)-N′-(2-trifluoro-methyl-phenyl)-guanidine 394

Microwave and Ultrasound Irradiation-Assisted Synthesis of Novel Disaccharide-Derived Arylsulfonyl Thiosemicarbazides 400

2007年 406

Synthesis of New Plant Growth Regulator:N-(fatty acid)O-aryloxyacetyl Ethanolamine 406

Synthesis,Bioactivity,Theoretical and Molecular Docking Study of 1-Cyano-N-substituted-cyclopropanecarboxamide as Ketol-acid Reductoisomerase Inhibitor 411

单嘧磺隆晶体-活性构象转换的分子动力学模拟 420

基于受体结构的AHAS抑制剂的设计、合成及生物活性 427

The Design,Synthesis,and Biological Evaluation of Novel Substituted Purines as HIV-1 Tat-TAR Inhibitors 431

酵母AHAS酶与磺酰脲类抑制剂作用模型的分子对接研究 444

2008年 450

High Throughput Screening Under Zinc-Database and Synthesis a Dialkylphos-phinic Acid as a Potential Kari Inhibitor 450

N-(4′-取代嘧啶-2′-基)-2-甲氧羰基-5-(取代)苯甲酰胺基苯磺酰脲化合物的合成及除草活性研究 453

Synthesis and Herbicidal Activity of Novel Sulfonylureas Containing Thiadiazol Moiety 465

The Outset Innovation of Agrochemicals in China 471

2009年 477

Quantitive-structure Activity Relationship(QSAR)Study of a New Heterocyclic Insecticides Using CoMFA and CoMSIA 477

Design,Synthesis,and Fungicidal Activity of Novel Analogues of Pyrrolnitrin 483

新型苯环5-(取代)苯甲酰胺基苯磺酰脲类化合物的比较定量构效关系研究 496

Regioselective Synthesis of Novel 3-Alkoxy(phenyl)thiophosphorylamido-2-(per-O-acetylglycosyl-1′-imino) Thiazolidine-4-one Derivatives from O-alkyl N4-glycosyl(thiosemicarbazido) Phosphonothioates 501

Synthesis,Herbicidal Activities and Comparative Molecular Field Analysis Study of Some Novel Triazolinone Derivatives 512

Synthesis,Antifungal Activities and 31D-QSAR Study of N-(5-substituted-1,3,4-thiadiazol-2-yl) Cyclopropanecarboxamides 526

Synthesis,Bioactivity and SAR Study of N′-(5-substituted-1,3,4-thiadiazol-2-yl)-N-cyclopropylformyl-thioureas as Ketol-acidReductoisomerase Inhibitors 535

Synthesis and Biological Activity of Novel 2,3-Dihydro-2-phenylsulfonyl-hydrazono-3-(2′,3′,4′,6′-tetra-O-acetyl-β-D-glucopyranosyl)thiazoles 546

4,5,6-三取代嘧啶苯磺酰脲类化合物的生物活性、分子对接与3D-QSAR关系研究 552

2010年 559

Synthesis, Crystal Structure and Insecticidal Activities of Novel Neonicotinoid Derivatives 559

区域选择性合成2-取代磺酰基亚肼基-3-全乙酰糖基-2, 3-二氢噻唑及其表征、生物活性研究 567

3位苯甲酰腙和亚氨基取代硫脲取代的吲哚满二酮衍生物的合成及对AHAS的抑制活性 573

Synthesis and Biological Activity of Some Novel Trifluoromethyl-Substituted 1,2,4-Triazole and Bis(1,2,4-Triazole) Mannich Bases Containing Piperazine Rings 578

Synthesis and Fungicidal Activity of Novel Aminophenazine-1-carboxylate Derivatives 594

High Throughput Receptor-based Virtual Screening under ZINC Database,Synthesis,and Biological Evaluation of Ketol-acid Reductoisomerase Inhibitors 618

2011年 627

Synthesis and Insecticidal Activities of Novel Analogues of Chlorantraniliprole Containing Nitro Group 627

Modulations of High-voltage Activated Ca2+ Channels in the Central Neurones of Spodoptera Exigua by Chlorantraniliprole 634

Synthesis,Structure and Biological Activity of Novel 1,2,4-Triazole Mannich Bases Containing a Substituted Benzylpiperazine Moiety 641

Design,Synthesis and Antifungal Activities of Novel Pyrrole Alkaloid Analogs 654

Synthesis and Insecticidal Evaluation of Novel N-Pyridylpyrazolecarboxamides Containing Different Substituents in the ortho-Position 675

Synthesis,Crystal Structure,Bioactivity and DFT Calculation of New Oxime Ester Derivatives Containing Cyclopropane Moiety 684

2012年 693

The Structure-activity Relationship in Herbicidal Monosubstituted Sulfonylureas 693

Synthesis,Crystal Structure and Biological Activities of Novel Anthranilic ( Isoph-thalic)Acid Esters 708

Synthesis and Evaluation of Novel Monosubstituted Sulfonylurea Derivatives as Antituberculosis Agents 716

基于Ugi反应的新型鱼尼丁受体杀虫剂的设计、合成及生物活性 736

Synthesis and Insecticidal Activities of Novel Anthranilic Diamides Containing Acylthiourea and Acylurea 746

Design,Synthesis and Biological Activities of Novel Anthranilic Diamide Insecticide Containing Trifluoroethyl Ether 760

Evaluation of the in Vitro and Intracellular Effiicacy of New Monosubstituted Sulfonylureas against Extensively Drug-resistant Tuberculosis 779

2013年 786

Synthesis and Insecticidal Evaluation of Novel N-Pyridylpyrazolecarboxamides Containing Cyano Substituent in the ortho-Position 786

N-[4-氯-2-取代氨基甲酰基-6-甲基苯基]-1-芳基-5-氯-3-三氟甲基-1 H-吡唑-4-甲酰胺的合成及生物活性 795

Synthesis,Insecticidal Activities,and SAR Studies of Novel Pyridylpyrazole Acid Derivatives Based on Amide Bridge Modification of Anthranilic Diamide Insecticides 805

Design,Synthesis and Structure-activity of N-Glycosyl-1-pyridyl-1H- pyrazole-5-carboxamide as Inhibitors of Calcium Channels 826

新型含三唑啉酮的磺酰脲类化合物的合成、晶体结构及除草活性研究 839

Design,Syntheses and Biological Activities of Novel Anthranilic Diamide Insecticides Containing N-Pyridylpyrazole 853

Synthesis and Biological Activities of Novel Anthranilic Diamides Analogues Containing Benzo[b]thiophene 865

附录 879

附录1论文总目录 879

附录2专利及著作目录 911

附录3历年指导的学生名单 915